SCHEMBL746591

SCHEMBL746591

CC(C)(C)c1ccc(CN(CCc2ccc(F)c(F)c2)C(=O)c2cc(Cl)cc3c2NCCC3)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
ESRRG P62508 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
NCOA1 Q15788 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
C5AR1 P21730 1/20 0.32
PPARG P37231 1/20 0.31
MAPK14 Q16539 1/20 0.31
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL747122 0.95 TP53 (0.33) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL748492 0.94 TP53 (0.33) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL751012 0.94 PARP1 (0.36) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL747648 0.93 PARP1 (0.36) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL747155 0.92 TP53 (0.38) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL748268 0.92 TP53 (0.38) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL745512 0.91 OPRM1 (0.34) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL747110 0.90 OPRM1 (0.34) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL748780 0.89 TP53 (0.35) PARP1TP53MAPTESRRGKDM4E
SCHEMBL748464 0.87 ALDH1A1 (0.37) MAPTKDM4EMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP claimed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US claimed
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed