SCHEMBL7471615

SCHEMBL7471615

[CH](Cc1ccncc1)Cc1ccco1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.38
KDM4E B2RXH2 3/20 0.38
MAPK1 P28482 2/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 6/20 0.38
GAA P10253 1/20 0.38
TP53 P04637 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KDM6B O15054 1/20 0.35
KDM4A O75164 1/20 0.35
KDM5C P41229 1/20 0.35
KDM4D Q6B0I6 1/20 0.35
KDM4C Q9H3R0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5495225 0.78 CYP3A4 (0.55) LMNAMAPK1ALDH1A1CYP1A2CYP3A4
SCHEMBL1255865 0.76 LOXL2 (0.43) LMNAKDM4EMAPK1HTTALDH1A1
SCHEMBL3659294 0.75
SCHEMBL7471622 0.73 ALDH1A1 (0.46) LMNAKDM4EMAPK1HTTALDH1A1
SCHEMBL6948750 0.72 CYP1A2 (0.54) LMNAKDM4EMAPK1HTTALDH1A1
SCHEMBL27881714 0.71 MEN1 (0.65) LMNAKDM4EMAPK1HTTALDH1A1
SCHEMBL8117581 0.71 POLB (0.54) MAPK1HTTALDH1A1GAANPC1
SCHEMBL4657208 0.70
SCHEMBL5616217 0.69 CYP1A2 (0.40) LMNAKDM4EMAPK1HTTALDH1A1
SCHEMBL7380489 0.68 CYP1A2 (0.48) ALDH1A1CYP1A2CYP2D6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871619-B1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMA (US) 2002-11-06 EP disclosed
US-6458959-B1 VIRICIDES AND ENZYME INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-10-01 US disclosed
US-6348477-B1 SUBSTITUTED PHENYL THIAZOLE DERIVATIVES AS VIRICIDES BOEHRINGER INGELHEIM(CANADA) LTD. (CA) 2002-02-19 US disclosed
US-6057451-A AMINOTHIAZOLE DERIVATIVES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-05-02 US disclosed