SCHEMBL7471622

SCHEMBL7471622

c1coc(CCCc2ccncc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
CYP3A4 P08684 3/20 0.46
ALOX15 P16050 1/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HRH1 P35367 2/20 0.44
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.41
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
NAAA Q02083 1/20 0.38
CYP1A2 P05177 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1255865 0.89 LOXL2 (0.43) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL7364038 0.82 ALDH1A1 (0.50) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL11060991 0.82 ALDH1A1 (0.61) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL28161942 0.79 ALDH1A1 (0.55) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL30814185 0.78 KMT2A (0.57) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL7094868 0.77 ALDH1A1 (0.67) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL351920 0.77 HRH1 (0.65) ALDH1A1CYP3A4TDP1HRH1HRH4
SCHEMBL7093157 0.75 ALDH1A1 (0.70) ALDH1A1CYP3A4ALOX15USP2HPGD
SCHEMBL31673871 0.75 HRH1 (0.62) ALDH1A1CYP3A4TDP1HRH1HRH4
SCHEMBL28055322 0.75 HRH1 (0.62) ALDH1A1CYP3A4TDP1HRH1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871619-B1 PHENYL THIAZOLE DERIVATIVES WITH ANTI HERPES VIRUS PROPERTIES BOEHRINGER INGELHEIM PHARMA (US) 2002-11-06 EP disclosed
US-6458959-B1 VIRICIDES AND ENZYME INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-10-01 US disclosed
US-6348477-B1 SUBSTITUTED PHENYL THIAZOLE DERIVATIVES AS VIRICIDES BOEHRINGER INGELHEIM(CANADA) LTD. (CA) 2002-02-19 US disclosed
US-6057451-A AMINOTHIAZOLE DERIVATIVES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-05-02 US disclosed