SCHEMBL7471903

SCHEMBL7471903

Cc1cc(Cc2ccc(F)cc2)ccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.46
PTGS2 P35354 2/20 0.46
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
TAAR1 Q96RJ0 3/20 0.38
LMNA P02545 2/20 0.37
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
CETP P11597 1/20 0.36
IDO1 P14902 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
HTT P42858 1/20 0.35
DAO P14920 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12789510 0.81 SKP2 (0.50) PTGS1PTGS2ESR1ESR2TAAR1
SCHEMBL7467558 0.81 ESR1 (0.44) ESR1ESR2TAAR1MAPTHPGD
SCHEMBL26464918 0.81 ESR1 (0.54) ESR1ESR2
SCHEMBL7468157 0.80 IDH1 (0.46) ESR1ESR2TAAR1ALDH1A1IDO1
SCHEMBL7465577 0.78 LTA4H (0.53) ESR1ESR2LMNAMAPTALDH1A1
SCHEMBL22482119 0.77 PTGS1 (0.46) PTGS1PTGS2ESR1ESR2TAAR1
SCHEMBL306113 0.77
SCHEMBL29421562 0.77
SCHEMBL16584850 0.77 LOXL2 (0.47) ESR1ESR2ALDH1A1LOXL2ACHE
SCHEMBL3901537 0.76 KDM4E (0.45) TAAR1MAPTALDH1A1IDO1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757986-B1 Arylpiperidine and arylpiperazine derivatives and drugs containing the same SUNTORY LTD (JP) 2002-06-12 EP disclosed
US-5723475-A Arylpiperidine and arylpiperazine derivatives and medicament containing the same SUNTORY LIMITED (JP) 1998-03-03 US disclosed
EP-0757986-A1 ARYLPIPERIDINE AND ARYLPIPERAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME SUNTORY LIMITED (JP) 1997-02-12 EP disclosed