SCHEMBL8564898

SCHEMBL8564898

COC(=O)COC1CCC(n2ccn(-c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)c2=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
PDK2 Q15119 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
PDE4B Q07343 1/20 0.31
PDE4D Q08499 1/20 0.31
ABHD6 Q9BV23 1/20 0.31
LPAR5 Q9H1C0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564893 1.00 ESR1 (0.39) ESR1ESR2PDK2HDAC6PDE4B
SCHEMBL8562237 0.87 ESR1 (0.39) ESR1ESR2HDAC6PDE4BPDE4D
SCHEMBL8562233 0.87 ESR1 (0.39) ESR1ESR2HDAC6PDE4BPDE4D
SCHEMBL7418940 0.82 ESR1 (0.42) ESR1ESR2HDAC6ABHD6
SCHEMBL7415517 0.77 DRD2 (0.43)
SCHEMBL7476926 0.76 DRD2 (0.32)
SCHEMBL7476930 0.76 DRD2 (0.32)
SCHEMBL8562566 0.74 DRD2 (0.35) LPAR5
SCHEMBL8562570 0.74 DRD2 (0.35) LPAR5
SCHEMBL7472118 0.73 ESR1 (0.41) ESR1ESR2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed