SCHEMBL7472648

SCHEMBL7472648

Cc1cc(NS(=O)(=O)c2n[nH]c(N)n2)ccc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.51
MAPT P10636 5/20 0.49
TP53 P04637 2/20 0.45
JAK2 O60674 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
IDH1 O75874 1/20 0.40
IDO1 P14902 1/20 0.38
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
CDC7 O00311 1/20 0.37
EEF2K O00418 1/20 0.37
PLK4 O00444 1/20 0.37
AURKA O14965 1/20 0.37
DYRK3 O43781 1/20 0.37
RPS6KA5 O75582 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
PIM1 P11309 1/20 0.37
PHKG2 P15735 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9247576 0.85 PKM (0.46) LMNAJAK2MEN1KMT2ACDK2
SCHEMBL9352767 0.81 CA1 (0.46) MAPTTP53MEN1KMT2AIDO1
SCHEMBL9352738 0.81 LMNA (0.47) LMNAMAPTTP53MEN1KMT2A
SCHEMBL5227239 0.75 GAA (0.50) MEN1KMT2AALDH1A1
SCHEMBL18856402 0.74 JAK2 (0.76) MAPTJAK2MEN1KMT2A
SCHEMBL9865806 0.70 SLC40A1 (0.38) LMNAKMT2AIDH1ALDH1A1
SCHEMBL27275299 0.70 LMNA (0.49) LMNAMAPTTP53MEN1KMT2A
SCHEMBL2034092 0.69 LMNA (0.52) LMNAMAPTIDH1IDO1RAB9A
SCHEMBL8313948 0.69 GAA (0.38) KMT2A
SCHEMBL9156934 0.69 LMNA (0.40) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724586-B1 PROCESS FOR PREPARING N-(2,6-DICHLORO-3-METHYLPHENYL)-5-7-DIHALO[1,2,4]TRIAZOLO[1,5A]PYRIMIDINE-2-SULFONAMIDE BY CYCLIZATION AND HALO-DEHYDROXYLATION DOW AGROSCIENCES LLC (US) 2002-01-23 EP disclosed
EP-0724586-A1 PROCESS FOR PREPARING N-(2,6-DICHLORO-3-METHYLPHENYL)-5-7-DIHALO 1,2,4]TRIAZOLO 1,5A]PYRIMIDINE-2-SULFONAMIDE BY CYCLIZATION AND HALO-DEHYDROXYLATION DOWELANCO (US) 1996-08-07 EP disclosed
EP-0444747-B1 Preparation of 5,7-dihydroxy-1,2,4-triazolo(1,5-a)-pyrimidine-2-sulfonanilides DOWELANCO (US) 1996-05-15 EP disclosed
WO-1995011246-A1 PROCESS FOR PREPARING N-(2,6-DICHLORO-3-METHYLPHENYL)-5-7-DIHALO[1,2,4]TRIAZOLO[1,5A]PYRIMIDINE-2-SULFONAMIDE BY CYCLIZATION AND HALO-DEHYDROXYLATION DOWELANCO (US) 1995-04-27 WO disclosed
EP-0444747-A2 Preparation of 5,7-dihydroxy-1,2,4-triazolo(1,5-a)-pyrimidine-2-sulfonanilides DOWELANCO (US) 1991-09-04 EP disclosed
US-5006656-A Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides DOWELANCO (US) 1991-04-09 US disclosed