SCHEMBL7474205

SCHEMBL7474205

CN(C(c1ccccc1)c1ccccc1)S(=O)(=O)CC#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.36
HRH1 P35367 2/20 0.36
ALDH1A1 P00352 4/20 0.36
TDP1 Q9NUW8 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36
GMNN O75496 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
PMP22 Q01453 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CCR5 P51681 1/20 0.36
MAOB P27338 1/20 0.35
TP53 P04637 1/20 0.33
HTT P42858 1/20 0.33
SRC P12931 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31374594 0.80 AOC3 (0.39) HTR2AHRH1ALDH1A1TDP1KDM4E
SCHEMBL7482504 0.75 CYP2C19 (0.51) ALDH1A1TDP1KDM4EMAPTKMT2A
SCHEMBL7306332 0.72 CYP2C19 (0.41) ALDH1A1TDP1KDM4EMAPTKMT2A
SCHEMBL7476459 0.71 ALDH1A1 (0.45) ALDH1A1MAPTKMT2ALMNAPOLB
SCHEMBL7308150 0.70 KCNA5 (0.44) ALDH1A1TDP1KDM4EMAPTKMT2A
SCHEMBL7317708 0.70 MMP3 (0.53) ALDH1A1TDP1KDM4EMAPTKMT2A
Water SCHEMBL28355612 0.69 CHRNA7 (0.56) HTR2AHRH1ALDH1A1TDP1KDM4E
SCHEMBL10564457 0.68 MAOB (0.42) HTR2AHRH1ALDH1A1TDP1KDM4E
SCHEMBL6638318 0.68 SRC (0.42) ALDH1A1TDP1KDM4EMAPTKMT2A
SCHEMBL10584824 0.67 HTR2A (0.41) HTR2AHRH1ALDH1A1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975594-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES PFIZER LTD (GB) 2002-09-18 EP disclosed
US-6281357-B1 HEADACHE THERAPY PFIZER INC 2001-08-28 US disclosed
EP-0975594-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES Pfizer Limited (GB) 2000-02-02 EP disclosed
WO-1999002493-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES PFIZER LIMITED (GB) 1999-01-21 WO disclosed