SCHEMBL7474824

SCHEMBL7474824

Nc1c2ccccc2nc(=O)c2sccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 6/20 0.53
ALDH1A1 P00352 6/20 0.53
KDM4E B2RXH2 6/20 0.53
HPGD P15428 4/20 0.53
GLA P06280 3/20 0.53
ACHE P22303 3/20 0.53
CASP1 P29466 2/20 0.53
CASP7 P55210 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
CHRM2 P08172 2/20 0.53
ADRA2A P08913 2/20 0.53
ADORA3 P0DMS8 2/20 0.53
CHRM1 P11229 2/20 0.53
SLC6A2 P23975 2/20 0.53
OPRM1 P35372 2/20 0.53
KCNH2 Q12809 2/20 0.53
NQO2 P16083 1/20 0.53
MAOA P21397 1/20 0.53
DRD1 P21728 1/20 0.53
ADRA1A P35348 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7382821 0.74 ADORA2A (0.46) HSD17B10ALDH1A1KDM4EHPGDGLA
SCHEMBL7474809 0.74 MAPT (0.44) HSD17B10ALDH1A1KDM4EHPGDGLA
SCHEMBL1008482 0.73 TLR8 (0.46) HSD17B10ALDH1A1KDM4EHPGDGLA
SCHEMBL27777002 0.73 TLR8 (0.50) HSD17B10ALDH1A1KDM4EHPGDGLA
Aminacrine SCHEMBL14999 0.72 HSD17B10 (1.00) HSD17B10ALDH1A1KDM4EHPGDGLA
Aminacrine SCHEMBL29354393 0.72 HSD17B10 (1.00) HSD17B10ALDH1A1KDM4EHPGDGLA
Aminacrine SCHEMBL18989123 0.70 HSD17B10 (0.95) HSD17B10ALDH1A1KDM4EHPGDGLA
Aminacrine SCHEMBL4907467 0.70 HSD17B10 (0.95) HSD17B10ALDH1A1KDM4EHPGDGLA
Aminacrine SCHEMBL635597 0.70 RAB9A (1.00) HSD17B10ALDH1A1KDM4EHPGDGLA
Aminacrine SCHEMBL14482032 0.70 HSD17B10 (0.95) HSD17B10ALDH1A1KDM4EHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000073313-A1 NEW TRICYCLIC AMIDINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2000-12-07 WO disclosed