SCHEMBL27777002

SCHEMBL27777002

Nc1nc2ccccc2c2sccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 8/20 0.50
TLR7 Q9NYK1 8/20 0.50
DCPS Q96C86 1/20 0.50
ADORA2A P29274 2/20 0.47
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 3/20 0.45
GLA P06280 2/20 0.45
CASP1 P29466 2/20 0.45
CASP7 P55210 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
CHRM2 P08172 1/20 0.45
ADRA2A P08913 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CHRM1 P11229 1/20 0.45
NQO2 P16083 1/20 0.45
MAOA P21397 1/20 0.45
DRD1 P21728 1/20 0.45
ACHE P22303 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7382821 0.86 ADORA2A (0.46) TLR8TLR7DCPSADORA2AKDM4E
SCHEMBL1008482 0.85 TLR8 (0.46) TLR8TLR7DCPSADORA2AKDM4E
SCHEMBL7474809 0.80 MAPT (0.44) TLR8TLR7DCPSADORA2AKDM4E
SCHEMBL11932906 0.79 MDM4 (0.42) CHRM2ADRA2AADORA3MAOADRD1
SCHEMBL1451457 0.78 MAOA (0.45) ADORA2AKDM4EALDH1A1MAOATDP1
SCHEMBL10169211 0.78 GPR3 (0.57) TLR8TLR7ADORA2AKDM4EALDH1A1
SCHEMBL28435353 0.76 NUDT1 (0.49) ADORA2AKDM4EALDH1A1HPGDADORA3
SCHEMBL27389038 0.74 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2MAPTDYRK1ACLK1
SCHEMBL29583288 0.73 DCPS (0.64) TLR8TLR7DCPSADORA2AKDM4E
SCHEMBL72801 0.73 DCPS (0.64) TLR8TLR7DCPSADORA2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528704-B Serine-threonine protein kinase and PARP modulators CYLENE PHARMACEUTICALS INC 2014-04-09 CN disclosed
CN-101528704-A Serine-threonine protein kinase and PARP modulators CYLENE PHARMACEUTICALS INC (US) 2009-09-09 CN disclosed