SCHEMBL7474848

SCHEMBL7474848

COC(=O)Cc1cn(Cc2ccc3oc(-c4nc(C(C)(C)C)cs4)cc3c2)c2ccc(OCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)cc12

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ICMT O60725 12/20 0.40
PPARD Q03181 4/20 0.38
PPARG P37231 3/20 0.38
PPARA Q07869 3/20 0.38
PLA2G2A P14555 2/20 0.37
F2RL3 Q96RI0 1/20 0.33
EGFR P00533 1/20 0.33
IGF1R P08069 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479941 0.93 PPARD (0.43) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL6598709 0.88 THRA (0.44) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL6599665 0.86 PLA2G2A (0.39) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL6598794 0.86 PLA2G2A (0.47) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL6601718 0.86 PLA2G2A (0.38) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL5810585 0.85 PLA2G2A (0.41) ICMTPPARDPPARGPPARAPLA2G2A
Acetic Acid SCHEMBL6598580 0.85 S1PR1 (0.40) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL5810419 0.84 PPARD (0.53) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL6597512 0.84 PLA2G2A (0.37) ICMTPPARDPPARGPPARAPLA2G2A
SCHEMBL6603373 0.84 PPARD (0.44) ICMTPPARDPPARGPPARAPLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1170009-A2 Thiazolybenzofuran derivatives and their use as SRS-A and leukotiene antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-01-09 EP disclosed
EP-0880519-A1 THIAZOLYLBENZOFURAN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-12-02 EP disclosed
WO-1997027190-A1 THIAZOLYLBENZOFURAN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-07-31 WO disclosed