SCHEMBL7475274

SCHEMBL7475274

Cc1ncccc1-n1cccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR1A P08908 1/20 0.40
HTR2C P28335 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
ALDH1A1 P00352 3/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MYC P01106 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NOS3 P29474 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28455570 0.80 IDO1 (0.53) GAACYP1A2CYP2C19ALDH1A1MAPT
SCHEMBL2185781 0.74 GAA (0.47) GAAKDM4EHTR2CALDH1A1POLB
SCHEMBL951160 0.74 GAA (0.44) GAAKDM4EHTR3EHTR3BHTR1A
SCHEMBL16302917 0.74 GAA (0.50) GAAKDM4EHTR3EHTR3BHTR1A
SCHEMBL20911925 0.74 HCRTR1 (0.40) KDM4EMAPTNPSR1MYCL3MBTL1
SCHEMBL2592089 0.74 ALDH1A1 (0.41) GAAKDM4EHTR3EHTR3BHTR1A
SCHEMBL29543738 0.74 MAPK1 (0.49) GAAKDM4EALDH1A1MAPTNPSR1
SCHEMBL2172244 0.74 MAPK1 (0.49) GAAKDM4EALDH1A1MAPTNPSR1
SCHEMBL10289389 0.74 HTR3E (0.40) GAAKDM4ECYP1A2CYP2C19HTR3E
SCHEMBL2625458 0.74 GAA (0.46) GAAKDM4ECYP1A2CYP2C19HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246799-A1 SUBSTITUTED PYRROLE MANNICH BASES TO COMBAT PAIN AND ALLERGIC REACTIONS Grünenthal GmbH (DE) 2002-10-09 EP disclosed
WO-2001047878-A1 SUBSTITUTED PYRROLE MANNICH BASES TO COMBAT PAIN AND ALLERGIC REACTIONS Grünenthal GmbH (DE) 2001-07-05 WO disclosed
WO-2001047882-A2 SUBSTANCE LIBRARY WHICH CAN BE OBTAINED BY REACTING ALDEHYDES WITH SECONDARY AMINES, ACID CHLORIDES AND NAPHTHOL, PYRROLE AND/OR INDOLE COMPOUNDS Grünenthal GmbH (DE) 2001-07-05 WO disclosed