SCHEMBL7476310

SCHEMBL7476310

COC(=O)c1ccc2c(c1)NC(=O)C(CC(O[SiH](C)C)C(C)(C)C)O2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.45
GAA P10253 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALOX5 P09917 1/20 0.42
HSD17B10 Q99714 4/20 0.39
ALOX15 P16050 2/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7475258 0.84 HSD17B10 (0.44) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL7470594 0.83 USP2 (0.53) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL8601457 0.83 USP2 (0.39) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL7463472 0.83 HSD17B10 (0.48) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL7464320 0.81 USP2 (0.38) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL7473281 0.80 MEN1 (0.38) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL7472425 0.80 PARP1 (0.45) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL7472196 0.79 KMT2A (0.44) USP2GAAMEN1KMT2AHSD17B10
SCHEMBL18581866 0.79 USP2 (0.56) USP2GAAMEN1KMT2AALOX5
SCHEMBL7476297 0.78 ALOX5 (0.42) USP2GAAMEN1KMT2AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869949-B1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO MCNEIL PHARM INC (US) 2002-12-18 EP disclosed
US-5854242-A Benzoxazine antimicrobial agents ORTHO PHARMACEUTICAL CORPORATION (US) 1998-12-29 US disclosed
EP-0869949-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-14 EP disclosed
US-5696117-A BACTERICIDE ORTHO PHARMACEUTICAL CORPORATION (US) 1997-12-09 US disclosed
WO-1997017333-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-05-15 WO disclosed