SCHEMBL7476430

SCHEMBL7476430

CCC(CC1CCOC1)c1cc(O)c(C(c2cccs2)C2CC2)c(=O)o1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ICMT O60725 2/20 0.36
NQO1 P15559 1/20 0.33
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
TSHR P16473 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435361 0.96 MEN1 (0.35) ICMTNQO1MEN1NPC1ALDH1A1
SCHEMBL7444332 0.95 ICMT (0.39) ICMTNQO1MEN1NPC1ALDH1A1
SCHEMBL7450971 0.89 NQO1 (0.34) NQO1HDAC3HDAC1HDAC2
SCHEMBL7449599 0.86
SCHEMBL6176061 0.85 CYP2C9 (0.39)
SCHEMBL7439058 0.85 MEN1 (0.34) NQO1MEN1NPC1ALDH1A1RAB9A
SCHEMBL7450139 0.85 HPGD (0.38) NQO1MEN1NPC1ALDH1A1KMT2A
SCHEMBL9286896 0.84 ICMT (0.35) ICMTNQO1MEN1NPC1ALDH1A1
SCHEMBL7435888 0.83 NQO1 (0.35) ICMTNQO1MEN1NPC1ALDH1A1
SCHEMBL7444011 0.83 HPGD (0.37) NQO1MEN1ALDH1A1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed