SCHEMBL7450971

SCHEMBL7450971

CCC(CC1CCOC1)c1cc(O)c(C(CC)c2cccs2)c(=O)o1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.34
CYP2C9 P11712 1/20 0.33
ERCC5 P28715 1/20 0.32
FEN1 P39748 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439058 0.95 MEN1 (0.34) NQO1CYP2C9FEN1HDAC3HDAC1
SCHEMBL7435888 0.94 NQO1 (0.35) NQO1CYP2C9HDAC1HDAC2
SCHEMBL7476430 0.89 ICMT (0.36) NQO1HDAC3HDAC1HDAC2
SCHEMBL7434821 0.85 CYP2C9 (0.31) CYP2C9
SCHEMBL9199709 0.85 MEN1 (0.33) NQO1CYP2C9FEN1HDAC3HDAC1
SCHEMBL7435361 0.85 MEN1 (0.35) NQO1FEN1HDAC3HDAC1HDAC2
SCHEMBL7444808 0.84 HPGD (0.39) NQO1
SCHEMBL9197378 0.83 ICMT (0.33) NQO1
SCHEMBL7444332 0.83 ICMT (0.39) NQO1
SCHEMBL7474994 0.83 HPGD (0.37) NQO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed