SCHEMBL7476501

SCHEMBL7476501

Cc1ccc(OC(C(=O)OC(C)(C)C)N2CCC2)cn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNB3 Q05901 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 4/20 0.34
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GPR119 Q8TDV5 3/20 0.32
LMNA P02545 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
GCK P35557 1/20 0.32
KCNH2 Q12809 1/20 0.32
DGAT1 O75907 2/20 0.32
GALR3 O60755 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413845 0.87 KMT2A (0.40) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL7413215 0.85 GPR119 (0.41) GPR119
SCHEMBL7478112 0.80
SCHEMBL7416015 0.80 KMT2A (0.34) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL7410349 0.78 CHRNB1 (0.38) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL7417332 0.78 JAK3 (0.35) GPR119
SCHEMBL7477219 0.78 SCN9A (0.31)
SCHEMBL7405119 0.78
SCHEMBL7413937 0.77 GPR119 (0.32) GPR119LMNA
SCHEMBL7412567 0.77 HRH3 (0.36) KMT2AMEN1GPR119LMNAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950057-B1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LAB (US) 2002-11-13 EP disclosed
US-6403575-B1 ANTI-INFLAMMATORIES ABBOTT LABORATORIES 2002-06-11 US disclosed
US-6133253-A NEURONAL CELL DEATH PREVENTORS AND ANTI-INFLAMMATORIES ABBOTT LABORATORIES (US) 2000-10-17 US disclosed