SCHEMBL7412567

SCHEMBL7412567

CC(C)(C)OC(=O)C(Oc1cnc(F)c(Cl)c1)N1CCC1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.36
CYP3A4 P08684 2/20 0.33
CYP3A5 P20815 2/20 0.33
SCN9A Q15858 8/20 0.33
GPR119 Q8TDV5 2/20 0.32
KMT2A Q03164 3/20 0.31
MEN1 O00255 2/20 0.31
SCN5A Q14524 1/20 0.31
MAPK1 P28482 1/20 0.31
LMNA P02545 1/20 0.31
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413937 0.87 GPR119 (0.32) GPR119LMNA
SCHEMBL7416015 0.83 KMT2A (0.34) HRH3GPR119KMT2AMEN1LMNA
SCHEMBL7411562 0.82 KMT2A (0.35) HRH3KMT2ALMNA
SCHEMBL7411225 0.82 KMT2A (0.35) HRH3KMT2ALMNA
SCHEMBL7478780 0.81 HRH3 (0.32) HRH3GPR119KMT2AMEN1LMNA
SCHEMBL7413845 0.81 KMT2A (0.40) HRH3KMT2AMEN1LMNA
SCHEMBL7407935 0.81 ABHD6 (0.35) CYP3A4CYP3A5GPR119
SCHEMBL8506871 0.80 ALDH1A1 (0.37) KMT2ALMNA
SCHEMBL8506868 0.80 ALDH1A1 (0.37) KMT2ALMNA
SCHEMBL7478135 0.80 SCN9A (0.33) HRH3SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950057-B1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LAB (US) 2002-11-13 EP disclosed
US-6403575-B1 ANTI-INFLAMMATORIES ABBOTT LABORATORIES 2002-06-11 US disclosed
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
US-6133253-A NEURONAL CELL DEATH PREVENTORS AND ANTI-INFLAMMATORIES ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
EP-0950057-A1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS Abbott Laboratories (US) 1999-10-20 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed
WO-1998025920-A1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LABORATORIES (US) 1998-06-18 WO disclosed