SCHEMBL7476595

SCHEMBL7476595

N=C(N)Nc1nc2c(s1)-c1nc(N)sc1CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.40
PIK3CB P42338 8/20 0.40
PIK3CG P48736 8/20 0.40
PIK3CD O00329 7/20 0.40
PI4KB Q9UBF8 3/20 0.40
PIK3C3 Q8NEB9 1/20 0.39
KCNH2 Q12809 1/20 0.36
ADORA1 P30542 1/20 0.35
FBP1 P09467 3/20 0.33
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
CFTR P13569 4/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MPI P34949 1/20 0.32
CCNT1 O60563 1/20 0.31
CDK1 P06493 1/20 0.31
CDK4 P11802 1/20 0.31
CCNB1 P14635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8073174 0.79 ADORA1 (0.37) PIK3CAPIK3CBPIK3CGPIK3CDPI4KB
Bromide SCHEMBL7480303 0.70 ALDH1A1 (0.56) PIK3CAPIK3CBPIK3CGPIK3CDCFTR
SCHEMBL3536095 0.69 TSHR (0.58) KDM4EALDH1A1MAPT
SCHEMBL13314772 0.69 TSHR (0.54) ADORA1ALDH1A1MAPT
SCHEMBL13314773 0.68 TSHR (0.56) APOBEC3AAPOBEC3GALDH1A1MAPT
SCHEMBL7478299 0.67 ALDH1A1 (0.34) PIK3CAPIK3CBPIK3CGPIK3CDPI4KB
SCHEMBL3537945 0.65 PDK1 (0.47) APOBEC3AAPOBEC3GCFTRALDH1A1MAPT
SCHEMBL3535533 0.65 CHKA (0.41) MAPT
Hydrochloric Acid SCHEMBL3538938 0.64 CHKA (0.40) MAPT
SCHEMBL7486311 0.64 POLB (0.33) PIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843681-B1 HETEROCYCLE-FUSED THIAZOLE DERIVATIVES YUNGJIN PHARMACEUTICAL CO LTD (KR) 2002-03-06 EP disclosed