SCHEMBL7477055

SCHEMBL7477055

COC(=O)CCN1CCC(N2CCN(c3ccc4c(c3)CCN(C)CC4)C2=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
F2 P00734 3/20 0.39
F10 P00742 3/20 0.39
MCHR1 Q99705 2/20 0.38
PRSS1 P07477 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PARP1 P09874 1/20 0.36
KHK P50053 1/20 0.35
HTR1A P08908 1/20 0.35
CHRM5 P08912 1/20 0.35
SLC6A2 P23975 1/20 0.35
HRH2 P25021 1/20 0.35
ADRA1D P25100 1/20 0.35
HTR1B P28222 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR1E P28566 1/20 0.35
HRH1 P35367 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473162 0.89 F10 (0.43) SMN1; SMN2F2F10MCHR1PRSS1
Hydrochloric Acid SCHEMBL8561724 0.88 F10 (0.43) SMN1; SMN2F2F10MCHR1PRSS1
SCHEMBL8562703 0.87 F2 (0.35) F2F10KHKSLC6A2USP30
SCHEMBL8562707 0.87 F2 (0.35) F2F10KHKSLC6A2USP30
Hydrochloric Acid SCHEMBL8561453 0.87 F2 (0.35) F2F10KHKSLC6A2USP30
SCHEMBL7474111 0.83 PARP1 (0.38) F2F10PARP1HRH3DRD2
SCHEMBL7474107 0.83 PARP1 (0.38) F2F10PARP1HRH3DRD2
Hydrochloric Acid SCHEMBL7476507 0.83 KHK (0.36) F2F10PRSS1ALDH1A1KHK
SCHEMBL7468477 0.82 DRD2 (0.35) F2F10MCHR1HRH1HRH3
SCHEMBL7468482 0.82 DRD2 (0.35) F2F10MCHR1HRH1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed