SCHEMBL7477103

SCHEMBL7477103

CC(CNS(=O)(=O)C(C)C)C1CC=C(c2ccccn2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 2/20 0.40
GRIA1 P42261 1/20 0.40
GRIA3 P42263 1/20 0.40
NPY5R Q15761 3/20 0.39
GRIA4 P48058 7/20 0.38
APLNR P35414 1/20 0.33
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
SMO Q99835 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470281 0.90 NPY5R (0.38) GRIA2GRIA1GRIA3NPY5RGRIA4
SCHEMBL7475999 0.78 GRIA1 (0.38) GRIA2GRIA1GRIA3GRIA4
SCHEMBL7478378 0.77 GRIA2 (0.41) GRIA2GRIA1GRIA3GRIA4
SCHEMBL7468611 0.76 GRIA2 (0.42) GRIA2GRIA1GRIA3NPY5RGRIA4
SCHEMBL7473863 0.76 GRIA2 (0.42) GRIA2GRIA1GRIA3GRIA4
SCHEMBL7470882 0.75 GRIA4 (0.50) GRIA2GRIA1GRIA3NPY5RGRIA4
SCHEMBL7467018 0.75 GRIA2 (0.62) GRIA2GRIA1GRIA3NPY5RGRIA4
SCHEMBL7473870 0.71 NPY5R (0.38) GRIA2GRIA1GRIA3NPY5RGRIA4
SCHEMBL7474813 0.71 GRIA2 (0.46) GRIA2GRIA1GRIA3GRIA4
SCHEMBL5877559 0.69 GRIA4 (0.68) GRIA2GRIA1GRIA3NPY5RGRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937708-B1 Sulphonamide derivatives LILLY CO ELI (US) 2002-12-18 EP disclosed
US-6362230-B1 ALZHEIMER'S DISEASE ELI LILLY AND COMPANY 2002-03-26 US disclosed
EP-0937708-A2 sulphonamide derivatives ELI LILLY AND COMPANY (US) 1999-08-25 EP disclosed