SCHEMBL7470281

SCHEMBL7470281

CC(CNS(=O)(=O)C(C)C)C1CC=C(c2ccc(-c3ccccn3)s2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 2/20 0.38
GRIA2 P42262 2/20 0.37
PKM P14618 1/20 0.37
GRIA1 P42261 1/20 0.37
GRIA3 P42263 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
GHSR Q92847 4/20 0.34
ALDH1A1 P00352 1/20 0.34
MMP13 P45452 1/20 0.34
CHRNA7 P36544 2/20 0.33
F2 P00734 1/20 0.33
ALOX5 P09917 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477103 0.90 GRIA2 (0.40) NPY5RGRIA2GRIA1GRIA3GRIA4
SCHEMBL7478378 0.79 GRIA2 (0.41) GRIA2GRIA1GRIA3GRIA4
SCHEMBL7473870 0.76 NPY5R (0.38) NPY5RGRIA2PKMGRIA1GRIA3
SCHEMBL7475999 0.76 GRIA1 (0.38) GRIA2GRIA1GRIA3GRIA4
SCHEMBL7470882 0.72 GRIA4 (0.50) NPY5RGRIA2GRIA1GRIA3GRIA4
SCHEMBL7468611 0.72 GRIA2 (0.42) NPY5RGRIA2GRIA1GRIA3GRIA4
SCHEMBL7473863 0.71 GRIA2 (0.42) GRIA2GRIA1GRIA3F2GRIA4
SCHEMBL7467018 0.70 GRIA2 (0.62) NPY5RGRIA2GRIA1GRIA3GRIA4
SCHEMBL7474813 0.69 GRIA2 (0.46) GRIA2GRIA1GRIA3GRIA4
SCHEMBL8611621 0.69 PKM (0.36) PKMKDM4ENPC1GLAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937708-B1 Sulphonamide derivatives LILLY CO ELI (US) 2002-12-18 EP disclosed
US-6362230-B1 ALZHEIMER'S DISEASE ELI LILLY AND COMPANY 2002-03-26 US disclosed
EP-0937708-A2 sulphonamide derivatives ELI LILLY AND COMPANY (US) 1999-08-25 EP disclosed