SCHEMBL7477456

SCHEMBL7477456

Cn1c(Cc2nc3cc(C#N)ccc3[nH]2)nc2ccc(C(=O)O)cc21

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 1/20 0.44
NPSR1 Q6W5P4 1/20 0.41
PIN1 Q13526 1/20 0.41
PPARG P37231 11/20 0.40
APEX1 P27695 1/20 0.39
LGALS8 O00214 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
RORC P51449 1/20 0.38
ACSL1 P33121 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7478557 0.85 NPSR1 (0.43) NPSR1PPARGAPEX1LGALS8ALDH1A1
SCHEMBL7481362 0.80 PIN1 (0.40) GLP1RPIN1
SCHEMBL7477294 0.74 APEX1 (0.44) NPSR1APEX1ALDH1A1MAPK1
SCHEMBL9063730 0.73 GRIN1 (0.51) PIN1GRIN1GRIN2B
SCHEMBL6172717 0.71 PPARG (0.53) GLP1RPPARGLGALS8
SCHEMBL4069583 0.71 PIN1 (0.49) PIN1GRIN1GRIN2BALDH1A1
SCHEMBL29281094 0.71 LGALS8 (0.55) PPARGLGALS8
Hydrochloric Acid SCHEMBL6170063 0.70 PPARG (0.54) GLP1RPPARGLGALS8
SCHEMBL7408823 0.70 F10 (0.59)
SCHEMBL7072284 0.70 KMT2A (0.45) ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000020400-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATING HEPATITIS C INFECTIONS AXYS PHARMACEUTICALS, INC. (US) 2000-04-13 WO disclosed