SCHEMBL7477463

SCHEMBL7477463

COC(=O)COc1cc(C#N)ccc1OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.52
PTGDR2 Q9Y5Y4 2/20 0.49
PTGER1 P34995 1/20 0.48
SMPD1 P17405 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
MAOB P27338 1/20 0.47
PPIA P62937 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HPGD P15428 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PKM P14618 1/20 0.45
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480705 0.87 PTGDR2 (0.64) MRGPRX4PTGDR2PTGER1MAOBPPIA
SCHEMBL31562503 0.85 ALDH1A1 (0.47) MRGPRX4SMPD1HDAC1HDAC8HDAC6
SCHEMBL6332053 0.83 MRGPRX4 (0.52) MRGPRX4PTGDR2PTGER1SMPD1HDAC1
SCHEMBL3490042 0.82 MAOB (0.57) MRGPRX4MAOBNPC1RAB9AHPGD
SCHEMBL6766128 0.82 MAOB (0.57) MRGPRX4SMPD1HDAC1HDAC8HDAC6
SCHEMBL1680776 0.81 MAOB (0.53) MRGPRX4PTGER1MAOBNPC1RAB9A
Acetoacetic Acid SCHEMBL27720127 0.80 KDM4E (0.51) MRGPRX4PTGDR2PTGER1MAOBPPIA
SCHEMBL1646681 0.80 MRGPRX4 (0.60) MRGPRX4PTGER1SMPD1HDAC1HDAC8
SCHEMBL31433068 0.79 GAA (0.49) PTGDR2NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL2327275 0.78 MRGPRX4 (0.53) MRGPRX4PTGDR2NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183235-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2002-03-06 EP disclosed
WO-2000071510-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2000-11-30 WO disclosed