SCHEMBL7477663

SCHEMBL7477663

CCCCCNc1nc(C)c(-c2ccc(OC)cc2CO)nc1OC

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 9/20 0.45
TLR7 Q9NYK1 5/20 0.37
TLR8 Q9NR97 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ACHE P22303 4/20 0.35
BCHE P06276 3/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7478779 0.88 CRHR1 (0.44) CRHR1TLR7TLR8ACHEBCHE
SCHEMBL5406607 0.82 CRHR1 (0.68) CRHR1
SCHEMBL6202450 0.80 CRHR1 (0.56) CRHR1TLR7
SCHEMBL7474607 0.79 CRHR1 (0.60) CRHR1
SCHEMBL7475201 0.79 CRHR1 (0.68) CRHR1
SCHEMBL7482544 0.78 CRHR1 (0.52) CRHR1TLR7TLR8
SCHEMBL7472049 0.78 CRHR1 (0.56) CRHR1TLR7
SCHEMBL6204586 0.77 USP8 (0.43) CRHR1TLR7ACHEBCHEALDH1A1
SCHEMBL6200464 0.77 TLR7 (0.42) CRHR1TLR7TLR8ALDH1A1
SCHEMBL7119050 0.77 CRHR1 (0.48) CRHR1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP claimed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO claimed