SCHEMBL7478236

SCHEMBL7478236

Oc1ccc2cc(CCC(O)Br)ccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
HCAR2 Q8TDS4 2/20 0.40
ALOX5 P09917 2/20 0.39
CYP3A4 P08684 2/20 0.38
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
HIF1A Q16665 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP17A1 P05093 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
ABL1 P00519 1/20 0.36
ABCB1 P08183 1/20 0.36
BCR P11274 1/20 0.36
GRIN2D O15399 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471821 0.83 CYP1A2 (0.45) CYP1A2ALOX5CYP3A4ESR1ESR2
SCHEMBL9125921 0.82 TYR (0.54) CYP1A2HCAR2ALOX5CYP3A4ESR1
SCHEMBL5505572 0.79 STAT3 (0.41) CYP1A2HCAR2ALOX5HSD17B10GRIN2D
SCHEMBL19012422 0.75 CA2 (0.60) CYP1A2HCAR2ALOX5CYP3A4ESR1
SCHEMBL5500720 0.75 STAT3 (0.40) CYP1A2ALOX5CYP3A4ESR1ESR2
SCHEMBL2921175 0.74 CYP1A2 (0.52) CYP1A2ALOX5CYP3A4ESR1ESR2
SCHEMBL12221232 0.74 ESR1 (0.52) CYP1A2HCAR2ALOX5CYP3A4ESR1
SCHEMBL17194110 0.73 GRIA2 (0.54) HCAR2ALOX15HIF1AHSD17B10TDP1
SCHEMBL16704739 0.73 GRIA2 (0.54) HCAR2ALOX15HIF1AHSD17B10TDP1
SCHEMBL14151517 0.73 CYP1A2 (0.46) CYP1A2HCAR2ALOX5CYP3A4ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed