SCHEMBL7478310

SCHEMBL7478310

CC(C(=O)NC(CC(=O)OC(C)(C)C)C(O)COC(=O)c1cccc(Cl)c1Cl)n1ccc2ccccc2c1=O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.38
ADRB1 P08588 4/20 0.38
ADRB3 P13945 4/20 0.38
CASP1 P29466 1/20 0.36
ELANE P08246 2/20 0.34
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
PSMB1 P20618 2/20 0.32
PSMB5 P28074 2/20 0.32
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL311815 0.92 CASP3 (0.36) ADRB2ADRB1ADRB3CASP1ELANE
SCHEMBL7472403 0.86 CASP1 (0.46) CASP1
SCHEMBL311567 0.77 CASP3 (0.50) CASP1ELANE
SCHEMBL10201581 0.70 ADRB2 (0.48) ADRB2ADRB1ADRB3CASP1KDM4E
SCHEMBL311493 0.68 ELANE (0.39) CASP1ELANE
SCHEMBL311492 0.68 ELANE (0.39) CASP1ELANE
SCHEMBL311790 0.67 CASP3 (0.62) CASP1
SCHEMBL10044272 0.67 CASP3 (0.62) CASP1
SCHEMBL87567 0.66 DDR1 (0.31) CASP1
SCHEMBL3908876 0.65 SYK (0.45) CASP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244626-A2 CASPASE INHIBITORS AND USES THEREOF Vertex Pharmaceuticals Incorporated (US) 2002-10-02 EP disclosed
WO-2001042216-A2 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2001-06-14 WO disclosed