SCHEMBL7478448

SCHEMBL7478448

C=Cc1cncc(OC[C@@H]2CCN2C(=O)OC(C)(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.42
CHRNA3 P32297 5/20 0.42
CHRNB4 P30926 4/20 0.42
CHRNA4 P43681 4/20 0.42
CHRNB1 P11230 3/20 0.41
CHRNB3 Q05901 3/20 0.41
CHRNA2 Q15822 1/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
DAPK3 O43293 1/20 0.37
ROCK2 O75116 1/20 0.37
PRKCG P05129 1/20 0.37
PIM1 P11309 1/20 0.37
RPS6KB1 P23443 1/20 0.37
AKT1 P31749 1/20 0.37
LIMK1 P53667 1/20 0.37
CDK5 Q00535 1/20 0.37
PRKCD Q05655 1/20 0.37
PAK1 Q13153 1/20 0.37
STK3 Q13188 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584401 0.94 CHRNB2 (0.47) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL7927287 0.87 CHRNB2 (0.44) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL6585964 0.86 CHRNB2 (0.60) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL7465912 0.86 CHRNB2 (0.57) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL7476340 0.86 DAPK3 (0.44) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL7475438 0.85 CHRNB2 (0.45) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL7475109 0.85 CHRNB2 (0.54) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL13335166 0.84 CHRNB2 (0.44) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL7474322 0.84 CHRNB2 (0.44) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1
SCHEMBL14941847 0.84 CHRNB2 (0.45) CHRNB2CHRNA3CHRNB4CHRNA4CHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950057-B1 3-PYRIDYL ENANTIOMERS AND THEIR USE AS ANALGESICS ABBOTT LAB (US) 2002-11-13 EP disclosed
US-6403575-B1 ANTI-INFLAMMATORIES ABBOTT LABORATORIES 2002-06-11 US disclosed
US-6133253-A NEURONAL CELL DEATH PREVENTORS AND ANTI-INFLAMMATORIES ABBOTT LABORATORIES (US) 2000-10-17 US disclosed