SCHEMBL7478704

SCHEMBL7478704

Cc1cnc2c(c1)C(=O)NC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.50
CDK5 Q00535 2/20 0.39
GSK3B P49841 2/20 0.39
PLK4 O00444 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
LCK P06239 1/20 0.39
CDK1 P06493 1/20 0.39
CSF1R P07333 1/20 0.39
PIM1 P11309 1/20 0.39
RPS6KB1 P23443 1/20 0.39
CDK2 P24941 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
MAPK8 P45983 1/20 0.39
CSNK1D P48730 1/20 0.39
MAPKAPK2 P49137 1/20 0.39
CLK2 P49760 1/20 0.39
GSK3A P49840 1/20 0.39
STK3 Q13188 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12108751 0.76 KMT2A (0.66) KMT2ACCR1CCR5CCR8PDK2
SCHEMBL6598757 0.76 KMT2A (0.66) KMT2ACCR1CCR5CCR8PDK2
SCHEMBL13151876 0.76 KMT2A (0.71) KMT2APIM1CCR1CCR5CCR8
SCHEMBL20672203 0.75 NPSR1 (0.41) KMT2ACDK5GSK3BPLK4PRKD3
SCHEMBL30029120 0.75 NPSR1 (0.41) KMT2ACDK5GSK3BPLK4PRKD3
SCHEMBL8661117 0.75 PPOX (0.50) KMT2ACDK5GSK3BPLK4PRKD3
SCHEMBL7485228 0.73 KMT2A (0.49) KMT2ACCR1CCR5CCR8ALDH1A1
SCHEMBL12191696 0.72 ALDH1A1 (0.44) KMT2ACDK5CCR1CCR5CCR8
SCHEMBL13544020 0.69 TDP1 (0.56) KMT2AGSK3BALDH1A1MAPTSMN1; SMN2
SCHEMBL13534041 0.69 KMT2A (0.38) KMT2ACDK5CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020120143-A1 Process for the preparation of 2,3-pyridinedicarboximides INTELLECTUAL PROPERTY DEPARTMENT, BASF AKTIENGESELLSCHAFT (DE) 2002-08-29 US disclosed
EP-0812842-B1 Process for the preparation of 5-(alkoxymethyl)-2,3-pyridine-dicarboximide compounds BASF AG (DE) 2002-03-27 EP disclosed
EP-0812843-B1 Process for the preparation of 2,3-pyridinedicarboximides BASF AG (DE) 2002-01-30 EP disclosed
US-6316629-B1 AS CHEMICAL INTERMEDIATES TO OBTAIN HERBICIDES AMERICAN CYANAMID CO. 2001-11-13 US disclosed
US-6034253-A CHEMICAL INTERMEDIATE FOR HERBICIDE AMERICA CYANAMID COMPANY (US) 2000-03-07 US disclosed
US-5905154-A CHEMICAL CONDENSATION OF OXIME WITH HALOMALEIMIDE FOR HERBICIDES AMERICAN CYANAMID COMPANY (US) 1999-05-18 US disclosed
US-5849916-A Process for the preparation of 2,3-pyridinedicarboximides AMERICAN CYANAMID COMPANY (US) 1998-12-15 US disclosed
EP-0812843-A2 Process for the preparation of 2,3-pyridinedicarboximides American Cyanamid Company (US) 1997-12-17 EP disclosed
EP-0812842-A2 Process for the preparation of 5-(alkoxymethyl)-2,3-pyridine-dicarboximide compounds American Cyanamid Company (US) 1997-12-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020120143-A1 Process for the preparation of 2,3-pyridinedicarboximides PNPO, CHRNA9, NAPRT KMT2A 1901/4885CDK5 829/4885GSK3B 3478/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.