SCHEMBL7478909

SCHEMBL7478909

C=Cn1c(C)c(C)c2cn[nH]c(=O)c21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 4/20 0.36
LMNA P02545 4/20 0.36
TSHR P16473 4/20 0.36
HSD17B10 Q99714 3/20 0.36
KDM4A O75164 1/20 0.36
TDP1 Q9NUW8 2/20 0.34
RECQL P46063 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
XDH P47989 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ADORA2A P29274 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRA1A P35348 1/20 0.33
RAB9A P51151 1/20 0.33
BLM P54132 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9742076 0.78 ALDH1A1 (0.44) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7475545 0.78 KDM4E (0.42) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7482128 0.71 ALDH1A1 (0.38) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7477781 0.71 KDM4E (0.47) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7479944 0.71 ALDH1A1 (0.41) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7479948 0.71 ALDH1A1 (0.41) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7476256 0.71 KDM4E (0.41) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7478732 0.70 KDM4E (0.39) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7478727 0.70 KDM4E (0.39) ALDH1A1KDM4ELMNATSHRHSD17B10
SCHEMBL7485703 0.70 KDM4E (0.41) ALDH1A1KDM4ELMNATSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed