SCHEMBL7482128

SCHEMBL7482128

Cc1c(C)n(C2CC2)c2c(=O)[nH]ncc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 5/20 0.36
HSD17B10 Q99714 3/20 0.36
LMNA P02545 3/20 0.36
TSHR P16473 3/20 0.36
KDM4A O75164 1/20 0.36
METAP2 P50579 1/20 0.36
CYP11B2 P19099 1/20 0.34
CYP1A2 P05177 4/20 0.33
CYP2C9 P11712 4/20 0.33
CYP2C19 P33261 4/20 0.33
CHRM4 P08173 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KMT2A Q03164 3/20 0.33
CYP3A4 P08684 3/20 0.32
CYP2D6 P10635 2/20 0.32
KCNH2 Q12809 2/20 0.32
POLB P06746 1/20 0.32
PIK3CA P42336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480350 0.93 GAA (0.37) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL9742076 0.77 ALDH1A1 (0.44) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL7476910 0.75 KDM4E (0.41) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL23123689 0.73 ALDH1A1 (0.38) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL7473946 0.72 TRPC5 (0.44) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL7478909 0.71 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL5237590 0.71 CYP1A2 (0.45) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL7474494 0.71 CYP1A2 (0.45) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL5237595 0.71 CYP1A2 (0.45) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL7477781 0.70 KDM4E (0.47) ALDH1A1KDM4EHSD17B10LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed