SCHEMBL7480071

SCHEMBL7480071

CC(C)(C)C(=O)CN1C(=O)C=NC(c2ccccn2)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 3/20 0.40
CCKAR P32238 1/20 0.40
RIPK1 Q13546 1/20 0.38
ALDH1A1 P00352 5/20 0.38
POLB P06746 1/20 0.35
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920133 0.76 ALDH1A1 (0.36) ALDH1A1
SCHEMBL7069964 0.74 FDFT1 (0.37) CCKBRALDH1A1POLBTHRB
SCHEMBL8548817 0.72 CCKBR (0.38) CCKBRCCKARALDH1A1
SCHEMBL8544961 0.66 CCKBR (0.61) CCKBRCCKAR
SCHEMBL8546357 0.66 CCKBR (0.61) CCKBRCCKAR
SCHEMBL4996686 0.66 CCKBR (0.61) CCKBRCCKAR
SCHEMBL4992176 0.65 CYP1A2 (0.59) CCKBRCCKARALDH1A1THRB
SCHEMBL8606321 0.63 ALDH1A1 (0.43) CCKBRCCKARALDH1A1POLBTHRB
SCHEMBL3910889 0.63 CCKBR (0.69) CCKBRCCKAR
SCHEMBL23352254 0.61 CYP1A2 (0.45) CCKBRCCKARRIPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951466-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS Elan Pharmaceuticals, Inc. (US) 1999-10-27 EP claimed
WO-1998028268-A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 1998-07-02 WO claimed