SCHEMBL7480246

SCHEMBL7480246

CCOC(=O)CC(NC(=O)CN1CCN(c2ccc3c(c2)CCN(C)CC3)C1=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 2/20 0.40
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
KCNH2 Q12809 2/20 0.37
ITGAV P06756 1/20 0.37
SLC6A2 P23975 2/20 0.36
HTR1A P08908 1/20 0.36
CHRM5 P08912 1/20 0.36
HRH2 P25021 1/20 0.36
ADRA1D P25100 1/20 0.36
HTR1B P28222 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469768 0.93 MAPT (0.41) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7474864 0.83 TMEM97 (0.39) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7468971 0.80 ITGB3 (0.42) ALDH1A1MAPTITGB3ITGA2BITGAV
Trifluoroacetic Acid SCHEMBL7481102 0.76 ITGB3 (0.48) ITGB3ITGA2BITGAV
SCHEMBL7479149 0.74 ITGB3 (0.40) ALDH1A1ITGB3ITGA2BDRD2DRD3
SCHEMBL7481505 0.74 DRD3 (0.41) ALDH1A1LMNAMAPTSMN1; SMN2DRD2
Hydrochloric Acid SCHEMBL7472463 0.73 DRD3 (0.42) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7590360 0.73 ITGB3 (0.41) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL7474275 0.73 ITGB3 (0.51) ALDH1A1MEN1KMT2ALMNAITGB3
SCHEMBL7407154 0.73 ITGB3 (0.47) ALDH1A1MEN1KMT2AITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed