SCHEMBL7468971

SCHEMBL7468971

CC(C)(C)OC(=O)N1CCc2ccc(N3CCN(CC(=O)NC(CC(=O)O)c4ccccc4)C3=O)cc2CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.42
ITGA2B P08514 4/20 0.42
NR1H2 P55055 1/20 0.39
ITGAV P06756 3/20 0.39
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
ESR2 Q92731 2/20 0.38
USP30 Q70CQ3 1/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 1/20 0.37
ATM Q13315 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7478252 0.85 ITGB3 (0.47) ITGB3ITGA2BITGAV
SCHEMBL7474864 0.84 TMEM97 (0.39) NR1H2ESR2ALDH1A1MAPTATM
SCHEMBL7419930 0.84 NR1H2 (0.49) NR1H2ESR2USP30ALDH1A1MAPT
Trifluoroacetic Acid SCHEMBL7481102 0.81 ITGB3 (0.48) ITGB3ITGA2BITGAV
SCHEMBL7480246 0.80 ALDH1A1 (0.40) ITGB3ITGA2BITGAVALDH1A1MAPT
SCHEMBL7473247 0.78 NR1H2 (0.47) NR1H2ESR2USP30ALDH1A1MAPT
SCHEMBL7481405 0.76 NR1H2 (0.42) ITGB3ITGA2BNR1H2ESR2ALDH1A1
SCHEMBL7465981 0.76 NR1H2 (0.40) ITGB3ITGA2BNR1H2ESR2ALDH1A1
SCHEMBL7468291 0.74 NR1H2 (0.38) NR1H2ESR2JAK2JAK3PTK2
Trifluoroacetic Acid SCHEMBL7480684 0.73 ITGB3 (0.49) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed