SCHEMBL7480993

SCHEMBL7480993

NC(=O)[C@@]12CN(Cc3ccccc3)C[C@@H]1c1ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.42
TSHR P16473 1/20 0.41
ARG1 P05089 1/20 0.41
ARG2 P78540 1/20 0.41
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP2D6 P10635 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
FUCA1 P04066 2/20 0.39
AMPD2 Q01433 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484214 0.87 SIGMAR1 (0.42) SIGMAR1ARG1ARG2SIRT1FUCA1
SCHEMBL7565511 0.84 SIGMAR1 (0.41) SIGMAR1ALDH1A1CYP2D6
SCHEMBL8019721 0.77 SIGMAR1 (0.43) SIGMAR1ARG1ARG2S1PR1S1PR5
SCHEMBL8019723 0.77 SIGMAR1 (0.43) SIGMAR1ARG1ARG2S1PR1S1PR5
SCHEMBL7491471 0.75 SIGMAR1 (0.47) SIGMAR1FUCA1OPRM1OPRK1GRIN1
SCHEMBL7491948 0.73 SIGMAR1 (0.46) SIGMAR1FUCA1OPRM1OPRK1
SCHEMBL8022956 0.73 SIGMAR1 (0.46) SIGMAR1FUCA1OPRM1OPRK1
SCHEMBL7491954 0.72 SIGMAR1 (0.43) SIGMAR1OPRM1OPRK1
SCHEMBL4994044 0.70 GAA (0.53) SIGMAR1TSHRALDH1A1CYP2D6AMPD2
SCHEMBL7484788 0.69 SIGMAR1 (0.47) SIGMAR1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1038873-B1 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake SERVIER LAB (FR) 2002-05-02 EP disclosed
US-6153640-A FOR TREATING DEPRESSION, PANIC ATTACKS, OBSESSIVE-COMPULSIVE DISORDERS, PHOBIAS, IMPULSIVE DISORDERS, DRUG ABUSE OR ANXIETY ADIR ET COMPAGNIE (FR) 2000-11-28 US disclosed
EP-1038873-A2 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake ADIR ET COMPAGNIE (FR) 2000-09-27 EP disclosed