SCHEMBL7565511

SCHEMBL7565511

COC(=O)[C@@]12CN(Cc3ccccc3)C[C@@H]1c1ccccc12

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.41
ADRA2A P08913 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2D6 P10635 1/20 0.41
MCHR1 Q99705 2/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480993 0.84 SIGMAR1 (0.42) SIGMAR1ALDH1A1CYP2D6
SCHEMBL7484214 0.79 SIGMAR1 (0.42) SIGMAR1ADRA2A
SCHEMBL8019723 0.74 SIGMAR1 (0.43) SIGMAR1ALDH1A1
SCHEMBL8019721 0.74 SIGMAR1 (0.43) SIGMAR1ALDH1A1
SCHEMBL3976439 0.73 OPRM1 (0.47) ALDH1A1CYP2D6BCHE
SCHEMBL19779330 0.73 OPRM1 (0.47) ALDH1A1CYP2D6BCHE
SCHEMBL10306091 0.73 OPRM1 (0.47) ALDH1A1CYP2D6BCHE
SCHEMBL28554966 0.73 S1PR5 (0.45) ALDH1A1CYP2D6MCHR1BCHEMAOB
SCHEMBL19779328 0.73 OPRM1 (0.47) ALDH1A1CYP2D6BCHE
SCHEMBL15416062 0.73 CYP2D6 (0.44) SIGMAR1ALDH1A1CYP2D6MCHR1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1038873-B1 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake SERVIER LAB (FR) 2002-05-02 EP disclosed
US-6153640-A FOR TREATING DEPRESSION, PANIC ATTACKS, OBSESSIVE-COMPULSIVE DISORDERS, PHOBIAS, IMPULSIVE DISORDERS, DRUG ABUSE OR ANXIETY ADIR ET COMPAGNIE (FR) 2000-11-28 US disclosed
EP-1038873-A2 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake ADIR ET COMPAGNIE (FR) 2000-09-27 EP disclosed