SCHEMBL7483350

SCHEMBL7483350

O=c1oc(CC2(Cc3cccs3)CC2)cc(O)c1C(c1cccs1)C1CC1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.34
ICMT O60725 2/20 0.33
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32
MC4R P32245 1/20 0.32
HTR2B P41595 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443227 0.90 LMNA (0.33) NQO1ICMTKMT2ALMNAPKM
SCHEMBL7438660 0.89 ALDH1A1 (0.31) KMT2AALDH1A1
SCHEMBL7445304 0.88 NQO1 (0.31) NQO1ICMT
SCHEMBL7448078 0.87 NQO1 (0.31) NQO1ICMT
SCHEMBL7449202 0.86 ICMT (0.38) NQO1ICMT
SCHEMBL7446268 0.85 HPGD (0.36) KMT2ALMNAMEN1NPC1ALDH1A1
SCHEMBL7444575 0.85 ICMT (0.35) NQO1ICMT
SCHEMBL7450257 0.84 ALDH1A1 (0.36) KMT2ALMNAMEN1ALDH1A1
SCHEMBL7447997 0.84 ICMT (0.33) NQO1ICMTKMT2AMEN1NPC1
SCHEMBL7481812 0.83 NQO1 (0.34) NQO1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed