SCHEMBL7484688

SCHEMBL7484688

Nc1cc(NCc2ccccc2Cl)cc2nc(-c3ccco3)nn12

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.52
MAPT P10636 2/20 0.52
ADORA2A P29274 6/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TP53 P04637 1/20 0.49
ADORA1 P30542 2/20 0.46
ADORA3 P0DMS8 1/20 0.44
ADORA2B P29275 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431721 0.85 ADORA2A (0.56) THRBMAPTADORA2ATP53ADORA1
SCHEMBL7708996 0.84 ADORA3 (0.51) THRBMAPTADORA2AADORA1ADORA3
SCHEMBL6872375 0.82 ADORA2A (0.60) THRBMAPTADORA2ASMN1; SMN2TP53
SCHEMBL7709116 0.81 ADORA2A (0.48) THRBMAPTADORA2ASMN1; SMN2TP53
SCHEMBL7711822 0.80 PDE2A (0.42) THRBMAPTTP53
SCHEMBL7703042 0.79 ADORA2A (0.52) THRBMAPTADORA2A
SCHEMBL7705858 0.79 MAPT (0.46) THRBMAPTTP53
SCHEMBL7703121 0.78 ADORA2A (0.62) THRBMAPTADORA2ASMN1; SMN2TP53
SCHEMBL7708919 0.77 ADORA2A (0.56) MAPTADORA2AADORA1ADORA3ADORA2B
SCHEMBL7705841 0.76 ADORA2A (0.56) ADORA2AADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP claimed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US claimed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO claimed
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed