SCHEMBL7709116

SCHEMBL7709116

Nc1cc(NCc2ccccc2Cl)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.48
GPR39 O43194 2/20 0.46
KCNN3 Q9UGI6 1/20 0.42
NPC1 O15118 5/20 0.41
RAB9A P51151 3/20 0.41
F2 P00734 2/20 0.40
F10 P00742 1/20 0.40
KLKB1 P03952 1/20 0.40
MAPT P10636 6/20 0.39
TP53 P04637 3/20 0.39
THRB P10828 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HTT P42858 2/20 0.39
PPP1CA P62136 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703131 0.85 ADORA2A (0.46) ADORA2AKCNN3NPC1RAB9AF2
SCHEMBL7708909 0.84 ADORA2A (0.52) ADORA2ANPC1F2F10KLKB1
SCHEMBL6870348 0.83 ADORA2A (0.56) ADORA2AMAPTTP53SMN1; SMN2LMNA
SCHEMBL7711822 0.82 PDE2A (0.42) KCNN3NPC1RAB9AMAPTTP53
SCHEMBL7484688 0.81 THRB (0.52) ADORA2AMAPTTP53THRBSMN1; SMN2
SCHEMBL7705858 0.81 MAPT (0.46) KCNN3NPC1RAB9AMAPTTP53
SCHEMBL7708776 0.77 ADORA2A (0.53) ADORA2ANPC1RAB9AMAPTTP53
SCHEMBL7428533 0.74 ADORA2A (0.60) ADORA2ANPC1RAB9AF2MAPT
SCHEMBL7708907 0.73 ADORA2A (0.52) ADORA2ANPC1RAB9AMAPTTP53
SCHEMBL7438035 0.73 ADORA2A (0.59) ADORA2ANPC1RAB9AF2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed