SCHEMBL7484802

SCHEMBL7484802

COc1cc(CC(=O)CO)ccc1O[Si](C)(C)C(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.61
HTT P42858 3/20 0.43
LMNA P02545 3/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 5/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
CA5A P35218 1/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
ABL1 P00519 1/20 0.41
RIN1 Q13671 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
LDHA P00338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21359165 0.86 DRD2 (0.64) DRD2HTTLMNANPC1GAA
SCHEMBL21882882 0.85 DRD2 (0.66) DRD2HTTLMNANPC1GAA
SCHEMBL21359049 0.85 DRD2 (0.63) DRD2HTTLMNANPC1GAA
SCHEMBL3119147 0.83 DRD2 (0.56) DRD2HTTLMNANPC1GAA
SCHEMBL21154904 0.83 LMNA (0.58) HTTLMNANPC1GAAKMT2A
SCHEMBL7532262 0.81 DRD2 (0.58) DRD2HTTLMNANPC1GAA
SCHEMBL6049298 0.81 DRD2 (0.57) DRD2KMT2AMEN1
SCHEMBL8520391 0.80 DRD2 (0.57) DRD2KMT2AMEN1LDHA
SCHEMBL21359392 0.79 DRD2 (0.55) DRD2LMNAGAAKMT2AMEN1
SCHEMBL3122490 0.79 DRD2 (0.58) DRD2GAAKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
US-6004977-A ANTIDEPRESSANTS, COGNITION ACTIVATORS, AND ALZHEIMER'S DISEASE TREATMENT HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP disclosed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO disclosed