SCHEMBL7486018

SCHEMBL7486018

N#CCNC(=O)C1(NC(=O)c2ccc(OCc3csc(N4CCN(C(=O)O)CC4)n3)cc2)CCCCC1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSB P07858 19/20 0.62
CTSS P25774 18/20 0.62
CTSL P07711 17/20 0.62
CTSK P43235 5/20 0.62
CTSD P07339 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6183676 0.91 CTSB (0.60) CTSBCTSSCTSLCTSKCTSD
SCHEMBL6184370 0.85 CTSB (0.85) CTSBCTSSCTSLCTSK
SCHEMBL6183485 0.77 CTSB (1.00) CTSBCTSSCTSLCTSK
SCHEMBL6184277 0.77 CTSB (0.79) CTSBCTSSCTSLCTSK
SCHEMBL6181770 0.75 CTSB (0.83) CTSBCTSSCTSLCTSK
SCHEMBL6183543 0.75 CTSB (1.00) CTSBCTSSCTSLCTSK
Trifluoroacetic Acid SCHEMBL6182305 0.74 CTSB (0.89) CTSBCTSSCTSLCTSK
SCHEMBL1118162 0.71 GPR119 (0.52)
SCHEMBL6182905 0.70 CTSK (0.61) CTSBCTSSCTSLCTSK
SCHEMBL4576707 0.70 CTSB (1.00) CTSBCTSSCTSLCTSKCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed