SCHEMBL7486177

SCHEMBL7486177

CC1(C)CCC(=O)c2c(COc3ccccc3)n[nH]c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
BRD4 O60885 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALPL P05186 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
PKM P14618 1/20 0.36
ALDH1A1 P00352 2/20 0.34
MMP2 P08253 1/20 0.34
MMP13 P45452 1/20 0.34
GRM5 P41594 1/20 0.34
PARP1 P09874 1/20 0.34
GAA P10253 2/20 0.33
LMNA P02545 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7485590 0.77 PARP1 (0.33) CYP1A2PARP1
SCHEMBL7480513 0.74 ATM (0.41) NPC1RAB9AALPLHPGDALDH1A1
SCHEMBL7485922 0.72 PARP1 (0.50) ALPLCYP3A4CYP2C9HPGDCYP2C19
SCHEMBL6162395 0.70 CYP1A2 (0.41) CYP1A2BRD4NPC1RAB9AGRM5
SCHEMBL7486190 0.68 POLL (0.39) ALPLCYP3A4HPGDALDH1A1GAA
SCHEMBL7487084 0.68 HTR7 (0.41) NPC1RAB9AALPLHPGDALDH1A1
SCHEMBL6167448 0.67 CYP1A2 (0.39) CYP1A2RAB9AALDH1A1GRM5SMN1; SMN2
SCHEMBL6163500 0.63 CYP1A2 (0.46) CYP1A2GRM5
SCHEMBL7485161 0.62 CYP17A1 (0.34) ALPL
SCHEMBL25261032 0.60 ALOX12 (0.42) CYP1A2NPC1RAB9AHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed