SCHEMBL7486190

SCHEMBL7486190

COc1cccc(OC)c1-c1n[nH]c2c1C(=O)CCC2(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLL Q9UGP5 1/20 0.39
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
HPGD P15428 3/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
GSK3B P49841 2/20 0.37
GSK3A P49840 1/20 0.37
CYP3A4 P08684 2/20 0.37
MAPT P10636 1/20 0.37
SRD5A1 P18405 1/20 0.36
SRD5A2 P31213 1/20 0.36
ALPL P05186 1/20 0.35
HTR2C P28335 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
TOP1 P11387 1/20 0.33
PDE4A P27815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484067 0.81 GAA (0.50) ALDH1A1HPGDGAAMAPTALPL
SCHEMBL7482218 0.80 GSK3A (0.41) POLLALDH1A1GAAGSK3BGSK3A
SCHEMBL7486143 0.75 LRRK2 (0.39) ALPL
SCHEMBL7482943 0.74 HSP90AA1 (0.39) ALDH1A1KDM4EHPGDMAPTTDP1
SCHEMBL7487084 0.74 HTR7 (0.41) ALDH1A1KDM4EHPGDALPL
SCHEMBL7490668 0.73 ALPL (0.65) ALDH1A1KDM4EHPGDGSK3BGSK3A
SCHEMBL7486177 0.68 CYP1A2 (0.41) ALDH1A1HPGDGAACYP3A4ALPL
SCHEMBL7485922 0.64 PARP1 (0.50) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL266254 0.63 KDM4E (0.56) POLLALDH1A1KDM4EHPGDGLA
SCHEMBL8736314 0.63 ALDH1A1 (0.56) POLLALDH1A1KDM4EHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed