SCHEMBL7486185

SCHEMBL7486185

CC(C)C1CC(=O)c2c(CC(O)C3CC3)n[nH]c2C1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.43
HSD17B10 Q99714 1/20 0.33
BUB1 O43683 2/20 0.32
ALPL P05186 1/20 0.32
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31418674 0.59 HCAR2 (0.40) HCAR2BUB1
SCHEMBL6164331 0.57 DHODH (0.34)
SCHEMBL17987539 0.56
SCHEMBL25344995 0.55 TP53 (0.36)
SCHEMBL8283553 0.55 HCAR2 (0.76) HCAR2
SCHEMBL26685314 0.54 SHBG (0.39)
SCHEMBL26242998 0.53 HCAR2 (0.42) HCAR2
SCHEMBL26251966 0.53 HCAR2 (0.42) HCAR2
SCHEMBL26251972 0.53 HCAR2 (0.42) HCAR2
SCHEMBL17372084 0.52 NOS3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed