SCHEMBL7486195

SCHEMBL7486195

O=C(Cc1cccc(-c2ccccn2)c1)N1CCC[CH]C(O)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.43
CTSK P43235 3/20 0.42
KDM5C P41229 3/20 0.41
KDM4C Q9H3R0 3/20 0.41
KDM2A Q9Y2K7 3/20 0.41
KDM3A Q9Y4C1 3/20 0.41
KDM6B O15054 2/20 0.41
NPY5R Q15761 1/20 0.40
FFAR1 O14842 1/20 0.39
ALDH1A1 P00352 3/20 0.39
ECE2 P0DPD6 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HTR1A P08908 1/20 0.38
HTR7 P34969 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSL P07711 2/20 0.38
CTSB P07858 2/20 0.38
CTSS P25774 2/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5105817 0.82 CTSK (0.49) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL5105755 0.80 CTSK (0.43) POLBCTSKFFAR1ALDH1A1ECE2
SCHEMBL5105814 0.79 DAGLB (0.39) CTSKFFAR1HTR1AHTR7CTSL
SCHEMBL6578142 0.77 CTSK (0.48) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL5099441 0.76 CTSK (0.49) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL6590094 0.73 CTSK (0.47) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL4691175 0.73 CTSK (0.47) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL7429714 0.73 CTSK (0.64) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL5098711 0.73 CTSK (0.64) POLBCTSKKDM5CKDM4CKDM2A
SCHEMBL6404534 0.73 CTSK (0.64) POLBCTSKKDM5CKDM4CKDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed