SCHEMBL7486376

SCHEMBL7486376

CC(C)(C)[Si](Oc1cccc2c1CCC(N)C2)(c1ccccc1)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.58
DRD3 P35462 7/20 0.58
HTR6 P50406 1/20 0.41
PLAU P00749 1/20 0.41
DRD4 P21917 4/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
ADRA1A P35348 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8078287 0.80 DRD2 (0.37) DRD2DRD3DRD4CHRM2CHRM1
SCHEMBL7718891 0.80 DRD2 (0.36) DRD2DRD3DRD4CHRM2CHRM1
SCHEMBL7487384 0.79 DRD2 (0.67) DRD2DRD3DRD4
SCHEMBL7713227 0.78 CYP19A1 (0.37) DRD2CHRM2CHRM1CHRM3
SCHEMBL7718886 0.76 MTNR1A (0.39) DRD2DRD3DRD4
Hydrochloric Acid SCHEMBL6824058 0.76 DRD2 (0.97) DRD2DRD3PLAUDRD4CHRM2
Hydrochloric Acid SCHEMBL3468007 0.76 DRD2 (0.97) DRD2DRD3PLAUDRD4CHRM2
Hydrochloric Acid SCHEMBL31672141 0.76 DRD2 (0.97) DRD2DRD3PLAUDRD4CHRM2
Hydrochloric Acid SCHEMBL6824054 0.76 DRD2 (0.97) DRD2DRD3PLAUDRD4CHRM2
SCHEMBL7485460 0.76 ACHE (0.42) ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842161-B1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2002-09-18 EP disclosed
EP-1213285-A2 4,5-dipheny-oxazole derivatives and their use as platelet aggregation inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-06-12 EP disclosed
US-6300344-B1 FOR THERAPEUTIC AND/OR PROPHYLACTIC TREATMENT OF ARTERIAL OBSTRUCTION, CEREBROVASCULAR DISEASE, HEPATIC CIRRHOSIS, ARTERIOSCLEROSIS, ISCHEMIC HEART DISEASE, RESTENOSIS AFTER PERCUTANEOUS TRANSLUMINAL CORONARY ANGIOPLASTY, HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-09 US disclosed
US-5972965-A USEFUL FOR INHIBITION OF PLATELET AGGREGATION, VASODILATION, ANTIHYPERTENSIVE ACTIVITY AND PROSTAGLANDIN AGONIST FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-26 US disclosed
EP-0842161-A1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-05-20 EP disclosed
WO-1997003973-A1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-06 WO disclosed