SCHEMBL7486500

SCHEMBL7486500

C=CCOc1c(N)cc2c(C)cc(=O)oc2c1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.51
ALDH1A1 P00352 7/20 0.51
HPGD P15428 5/20 0.51
MAPT P10636 3/20 0.51
GAA P10253 5/20 0.50
L3MBTL1 Q9Y468 2/20 0.45
LMNA P02545 4/20 0.44
HTT P42858 2/20 0.44
GLA P06280 2/20 0.43
MAOA P21397 2/20 0.42
MAPK1 P28482 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR2C P28335 1/20 0.42
ADORA2A P29274 1/20 0.42
HSD17B10 Q99714 5/20 0.41
GFER P55789 1/20 0.41
TSHR P16473 1/20 0.41
MAOB P27338 2/20 0.40
UBE2N P61088 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7475095 0.81 KDM4E (0.47) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL4390489 0.76 KDM4E (0.79) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL29116625 0.75 KDM4E (0.77) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL7824982 0.70 LMNA (0.62) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL11313571 0.68 KDM4E (0.66) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL11309411 0.68 KDM4E (1.00) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL6898974 0.68 KDM4E (0.70) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL660817 0.67 ALDH1A1 (0.80) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL5312406 0.67 KDM4E (0.68) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL6865603 0.67 KDM4E (0.64) KDM4EALDH1A1HPGDMAPTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144417-B1 4'-SUBSTITUTED-4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABOR INC (US) 2002-09-04 EP disclosed
EP-1144417-A1 4'-SUBSTITUTED-4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2001-10-17 EP disclosed
US-6177424-B1 ANTIPROLIFERATIVE AGENTS, MICROBIOCIDES, ANTISEPTICS HEINDEL NED D (US) 2001-01-23 US disclosed
WO-2000032603-A1 4'-SUBSTITUTED-4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2000-06-08 WO disclosed