SCHEMBL7487153

SCHEMBL7487153

O=Cc1c[nH]c2cc(Cc3ccccc3)ccc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.57
IMPDH2 P12268 1/20 0.57
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MAPT P10636 1/20 0.51
PLG P00747 1/20 0.49
PLAU P00749 1/20 0.49
FEN1 P39748 1/20 0.46
PIM1 P11309 1/20 0.43
PIM3 Q86V86 1/20 0.43
PIM2 Q9P1W9 1/20 0.43
GABRA1 P14867 4/20 0.43
GABRB2 P47870 4/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GPR17 Q13304 1/20 0.42
GABRB1 P18505 1/20 0.41
GABRA3 P34903 1/20 0.41
CCNT1 O60563 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8746137 0.88 CYP2A6 (0.57) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL2279626 0.87 PLG (0.47) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL29955610 0.85 CYP2A6 (0.51) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL6819310 0.81 CYP2A6 (0.58) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL29957436 0.81 CYP2A6 (0.58) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL23725271 0.81 CYP2A6 (0.63) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL1418239 0.79 IMPDH2 (0.61) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL29951517 0.79 IMPDH2 (0.61) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL2535062 0.78 CYP2A6 (0.61) CYP2A6IMPDH2ALDH1A1KDM4EMAPT
SCHEMBL8746106 0.77 CYP2A6 (0.56) CYP2A6IMPDH2ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1226141-A1 HETEROCYCLIC SUBSTITUTED PYRAZOLONES CEPHALON, INC. (US) 2002-07-31 EP disclosed
WO-2001032653-A1 HETEROCYCLIC SUBSTITUTED PYRAZOLONES CEPHALON, INC. (US) 2001-05-10 WO disclosed