SCHEMBL7488641

SCHEMBL7488641

CCCCCCc1n[c]c2ncn(C)c2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.34
ADORA2B P29275 3/20 0.34
ADORA1 P30542 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
XDH P47989 1/20 0.33
TLR7 Q9NYK1 2/20 0.33
KCNH2 Q12809 1/20 0.33
SPNS2 Q8IVW8 1/20 0.32
CHRM2 P08172 2/20 0.32
CHRM4 P08173 2/20 0.32
CHRM5 P08912 2/20 0.32
CHRM1 P11229 2/20 0.32
CHRM3 P20309 2/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7492084 0.99 ADORA2A (0.35) ADORA2AADORA2BADORA1ADORA3XDH
SCHEMBL7487478 0.94 ADORA2A (0.34) ADORA2AADORA2BADORA1ADORA3XDH
SCHEMBL7489579 0.90 ADORA2A (0.32) ADORA2AADORA2BADORA1PDE4APDE4B
SCHEMBL7492011 0.77 CYP19A1 (0.40) ADORA2BTLR7
SCHEMBL7492889 0.77 CHRM2 (0.34) ADORA2BKCNH2SPNS2CHRM2CHRM4
SCHEMBL7488243 0.76 ADORA2B (0.40) ADORA2AADORA2BTLR7
SCHEMBL7486698 0.76 TSHR (0.41) ADORA2AADORA2BADORA1KCNH2KDM4E
SCHEMBL7488311 0.76 TSHR (0.41) ADORA2AADORA2BADORA1KCNH2KDM4E
SCHEMBL7492422 0.75 CHRM2 (0.32) ADORA2AADORA2BADORA1ADORA3KCNH2
SCHEMBL7491743 0.74 TSHR (0.41) ADORA2AADORA2BADORA1KCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915093-B1 AMIDE DERIVATIVES OTSUKA PHARMA CO LTD (JP) 2002-11-27 EP disclosed
US-6166016-A Amide derivatives OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2000-12-26 US disclosed
EP-0915093-A1 AMIDE DERIVATIVES OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1999-05-12 EP disclosed