SCHEMBL7488793

SCHEMBL7488793

CC(=O)Nc1ccc2[nH]c(=O)c(=O)n(C3CCCCC3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.56
OPRL1 P41146 5/20 0.56
OPRD1 P41143 5/20 0.51
OPRK1 P41145 5/20 0.51
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.51
PSMB8 P28062 1/20 0.48
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
OGFRL1 Q5TC84 1/20 0.45
PIK3CA P42336 1/20 0.44
MTOR P42345 1/20 0.44
PRKDC P78527 1/20 0.44
ERCC1 P07992 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17335974 0.79 ERCC1 (0.62) OPRM1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7476479 0.77 OPRL1 (0.65) OPRM1OPRL1OPRD1OPRK1KDM4E
SCHEMBL9395829 0.76 OPRM1 (0.64) OPRM1OPRL1OPRD1OPRK1
SCHEMBL8607620 0.75 ALDH1A1 (0.46) OPRM1OPRL1OPRD1OPRK1KDM4E
SCHEMBL8609111 0.74 PSMB8 (0.53) KDM4EALDH1A1HPGDHSD17B10PSMB8
SCHEMBL1270635 0.74 OPRM1 (0.74) OPRM1OPRL1OPRD1OPRK1OGFRL1
SCHEMBL30910142 0.73 OPRL1 (0.86) OPRM1OPRL1OPRD1OPRK1
SCHEMBL26092381 0.73 OPRL1 (0.86) OPRM1OPRL1OPRD1OPRK1
SCHEMBL1271514 0.73 OPRL1 (0.64) OPRM1OPRL1OPRD1OPRK1KDM4E
SCHEMBL1271664 0.71 OPRM1 (0.74) OPRM1OPRL1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799224-B1 QUINOXALINES AND DRUGS PREPARED THEREFROM BASF AG (DE) 2002-04-17 EP disclosed
US-5852017-A 2,3(1H,4H)-quinoxalinediones BASF AKTIENGESELLSCHAFT (DE) 1998-12-22 US disclosed
US-5849743-A Quinoxalines and drugs prepared therefrom BASF AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed
EP-0572852-B1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF AG (DE) 1998-10-21 EP disclosed
US-5714489-A 2,3(1H,4H)quinoxalinedione BASF AKTIENGESELLSCHAFT (DE) 1998-02-03 US disclosed
EP-0799224-A1 NOVEL QUINOXALINES AND DRUGS PREPARED THEREFROM BASF AKTIENGESELLSCHAFT (DE) 1997-10-08 EP disclosed
WO-1996019476-A1 NOVEL QUINOXALINES AND DRUGS PREPARED THEREFROM BASF AKTIENGESELLSCHAFT (DE) 1996-06-27 WO disclosed
EP-0572852-A1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF Aktiengesellschaft (DE) 1993-12-08 EP disclosed