SCHEMBL7489147

SCHEMBL7489147

C=CCc1c(F)cc(F)cc1Oc1cc(F)cc(F)c1CC=C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.33
ALDH1A1 P00352 1/20 0.31
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7494741 0.70 GABRA1 (0.34) POLB
SCHEMBL17748186 0.67
SCHEMBL17681681 0.67
SCHEMBL10986339 0.66 XDH (0.31) POLBALDH1A1PPARGPPARD
SCHEMBL23699844 0.65 TNKS (0.30)
SCHEMBL1624906 0.65 TDP1 (0.48) POLBALDH1A1PPARGPPARDPPARA
SCHEMBL18094957 0.65 DPP4 (0.42) ALDH1A1
SCHEMBL7494750 0.64 CYP3A4 (0.49) POLBALDH1A1PPARGPPARDPPARA
SCHEMBL10751466 0.64 CYP3A4 (0.53) POLBALDH1A1PPARGPPARDPPARA
SCHEMBL10989483 0.64 XDH (0.35) ALDH1A1PPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173170-A4 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2002-05-29 EP disclosed
EP-1173170-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-01-23 EP disclosed
US-6265434-B1 ANTIINFLAMMATORY AGENTS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000059503-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed