SCHEMBL7489274

SCHEMBL7489274

COc1cc(-c2nn(C)c(C#N)c2Cl)c(F)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 6/20 0.38
HSP90AA1 P07900 6/20 0.38
SRC P12931 2/20 0.36
PDE10A Q9Y233 3/20 0.36
PDE2A O00408 2/20 0.36
PPOX P50336 1/20 0.33
USP8 P40818 1/20 0.32
USP7 Q93009 1/20 0.32
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
KCNH2 Q12809 1/20 0.31
PRKDC P78527 1/20 0.31
EIF2AK3 Q9NZJ5 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
CCR6 P51684 1/20 0.31
CACNA1B Q00975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7690601 0.89 HSP90AB1 (0.39) HSP90AB1HSP90AA1SRCPDE10APDE2A
SCHEMBL7819187 0.83 PPOX (0.36) PPOX
SCHEMBL7811968 0.83 NPC1 (0.31) RAB9A
SCHEMBL7818695 0.82 SLC34A1 (0.30) RAB9A
SCHEMBL7811612 0.82 AR (0.34) PDE10A
SCHEMBL5398257 0.80 CYP1A2 (0.35) HSP90AB1HSP90AA1PDE10APDE2APPOX
SCHEMBL7686734 0.77 HSP90AB1 (0.49) HSP90AB1HSP90AA1SRCPDE10APDE2A
SCHEMBL6295368 0.77 PDE10A (0.33) HSP90AB1HSP90AA1SRCPDE10APDE2A
SCHEMBL9530563 0.77 PTGS2 (0.39) PDE10APDE2APPOXEIF2AK3ALDH1A1
SCHEMBL7487729 0.76 MAPT (0.41) PPOXALDH1A1MAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0769008-B1 PYRAZOLE DERIVATIVES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2002-05-22 EP disclosed
US-6083881-A Pyrazole derivatives as herbicides NOVARTIS CORPORATION (US) 2000-07-04 US disclosed
EP-0769008-A1 PYRAZOLE DERIVATIVES AS HERBICIDES Novartis AG (CH) 1997-04-23 EP disclosed
WO-1996001254-A1 PYRAZOLE DERIVATIVES AS HERBICIDES CIBA-GEIGY AG (CH) 1996-01-18 WO disclosed